Glossary of Terms

Plain-English explanations of scientific terms you’ll see across OncoForge.

•OH (Hydroxyl Radical)

One of the most reactive ROS—very damaging but very short-lived.

Also appears as: OH, hydroxyl radical

5

5-LOX (5-Lipoxygenase)

An enzyme that makes inflammatory signals (leukotrienes) which may support tumor growth.

Also appears as: ALOX5, 5LOX, 5 lipoxygenase

A

AKT (Protein Kinase B)

A survival signal inside cells. When overactive (common in cancer), it pushes growth and resists cell death. Many agents try to turn it down.

Also appears as: PKB, AKT1, AKT2, AKT3

ALDH (Aldehyde Dehydrogenase)

Detox enzymes; high ALDH activity can mark stem-like tumor cells in some cancers.

Also appears as: aldehyde dehydrogenase

AMPK

The cell’s fuel gauge. When switched on, it generally slows growth pathways like mTOR.

Also appears as: AMP-activated protein kinase

Angiogenesis

The building of new blood vessels. Tumors hijack this process to feed themselves. Anti-angiogenic therapies try to cut off that blood supply.

Also appears as: neovascularization, VEGF signaling

Anti-Proliferative

Slows or stops cells from multiplying.

Also appears as: antiproliferative

Antioxidant

Reduces oxidative stress. Timing around treatments can matter.

Apoptosis

A built-in, tidy self-destruct program for damaged cells. Many anticancer therapies try to switch this back on in tumor cells so they die cleanly.

Also appears as: programmed cell death, caspase-mediated cell death

Autophagy

Cellular recycling. It can help cells survive stress or, in some settings, lead to cell death.

Also appears as: macroautophagy

B

Bcl-2

A “stay alive” protein. High levels can help cancer cells resist cell death.

Also appears as: BCL2 family

Bioavailability

How much of a dose actually reaches the bloodstream and the target.

C

Cachexia

Cancer-related wasting—loss of weight and muscle with metabolic changes.

Caspase

A family of enzymes that carry out apoptosis once it’s been triggered.

Also appears as: caspases

Checkpoint Inhibitor

Immunotherapy drugs that take the brakes off T-cells (PD-1/PD-L1 or CTLA-4).

Also appears as: ICI, immune checkpoint inhibitor

Chelator

A metal-binding compound (e.g., for iron or copper) that can alter redox and drug actions.

Also appears as: metal chelator, chelation

Chemo Sensitivity

How strongly a tumor responds to a chemo drug. “Sensitizers” try to boost this response.

Also appears as: chemosensitivity, chemo-sensitivity

Chemosensitizer

Makes tumor cells more responsive to chemotherapy.

Also appears as: chemosensitization

Complex I (NADH Dehydrogenase)

The first big enzyme in the mitochondrial energy chain—targeted by some metabolic drugs.

Also appears as: Complex-I, CI, NADH dehydrogenase

COX-2

An inflammation enzyme that makes prostaglandins; frequently elevated in tumors.

Also appears as: PTGS2

CSC (Cancer Stem Cells)

A small, stubborn sub-group that can resist therapy and restart tumors.

Also appears as: cancer stem-like cells

CTL (Cytotoxic T Lymphocyte)

A T-cell that directly kills virus-infected or tumor cells.

Also appears as: CD8 T cell, killer T cell, cytotoxic T-cell

CTLA-4

Another T-cell brake that checkpoint drugs can target.

Also appears as: CTLA4

CYP1A1

A drug-metabolizing enzyme induced by some plant compounds and pollutants.

Also appears as: cytochrome P450 1A1, P450 1A1

CYP3A4

A liver enzyme that processes many drugs. Interactions can raise or lower drug levels.

Also appears as: cytochrome P450 3A4, P450 3A4

Cytostatic

Slows or stops cell growth rather than killing cells outright.

Cytotoxic

Directly kills cells.

D

DC (Dendritic Cells)

Key coaches of the immune system. They present tumor pieces to T-cells to kick off attacks.

Also appears as: dendritic, dendritic cells

DNA Intercalation

When flat molecules slide between DNA bases and jam copying or reading.

Also appears as: DNA intercalate, intercalator

DNMT (DNA Methyltransferase)

Adds methyl tags to DNA. DNMT inhibitors can lift certain gene silencing.

Also appears as: DNA methyltransferase

E

EGFR

A growth receptor on cell surfaces. When it’s too active, it can drive tumor growth.

Also appears as: ERBB1

EMT (Epithelial–Mesenchymal Transition)

A shift that makes tumor cells more mobile and invasive.

Endorphin

Natural “feel-good” chemicals that help with pain and well-being.

ER Stress (Endoplasmic Reticulum Stress)

When the cell’s protein-folding factory is overloaded, triggering stress responses that can end in cell death.

Also appears as: ER-Stress, unfolded protein response, UPR

ETC Bypass (Electron Transport Chain Bypass)

Rerouting electrons around parts of the mitochondrial chain to keep energy or redox flowing.

Also appears as: electron transport chain bypass

F

Ferroptosis

A form of cell death driven by iron and lipid oxidation—different from apoptosis.

Fibrin

A mesh-like clotting protein. Tumors can use fibrin to shield themselves.

Fucoidan

A sulfated fiber from brown seaweed with immune-modulating and investigational anti-tumor effects.

G

Galectin-3

A sugar-binding protein tied to fibrosis, immune tone, and spread (metastasis).

Glucose

Main sugar fuel for cells. Many tumors consume lots of it.

Glycolysis

The pathway that breaks down glucose for quick energy and building blocks—often dialed up in tumors.

GPx (Glutathione Peroxidase)

Antioxidant enzymes that detox peroxides using glutathione.

Also appears as: glutathione peroxidase

GSH (Glutathione)

A major antioxidant that helps detoxify cells and maintain redox balance.

Also appears as: glutathione

GSTP1

A detox enzyme (glutathione S-transferase pi) linked to drug resistance.

Also appears as: glutathione S-transferase pi

H

HA (Hyaluronic Acid)

A water-holding sugar in the tissue space around cells. Lots of HA can make tumors stiffer and harder to reach with drugs.

Also appears as: Hyaluronan, HA

HAS2/3 (Hyaluronan Synthase 2/3)

Enzymes that make hyaluronic acid. When very active, they can thicken the tumor matrix and hinder blood flow.

Also appears as: HAS2, HAS3, hyaluronan synthase

HDAC (Histone Deacetylase)

An epigenetic “tightener.” HDAC inhibitors can re-open silenced genes and slow growth.

Hedgehog Pathway

A developmental signal route (SMO/GLI) that some tumors co-opt for growth.

Also appears as: Sonic hedgehog, SHH, SMO, GLI

HER2 (ERBB2)

A growth receptor that’s amplified in some cancers (like breast and gastric). Targeted drugs can block it.

Also appears as: ERBB2, HER-2

HIF-1α (Hypoxia-Inducible Factor 1-alpha)

A low-oxygen “sensor” that helps tumors adapt when oxygen is scarce. It can drive new blood-vessel growth and make treatment harder.

Also appears as: HIF-1a, HIF1A, HIF

HRD (Homologous Recombination Deficiency)

A DNA-repair weakness that can sensitize tumors to PARP inhibitors and certain chemo.

HSP27 (Heat Shock Protein 27)

A stress-response helper protein that can protect tumor cells from death signals.

Also appears as: HSP 27, HSPB1

Hypoxia

Low oxygen—common inside tumors. It changes metabolism and can blunt treatment.

L

Lectin

A protein that sticks to sugars; some affect immunity or how cells stick and move.

M

Macrophage Activator

A compound that wakes up macrophages (innate immune cells) so they better recognize and attack threats.

Also appears as: macrophage activation

MAPK/ERK

A growth pathway downstream of RAS/RAF. It’s frequently overactive in cancer.

Also appears as: ERK, RAS–RAF–MEK–ERK, MAPK

Mcl-1

A BCL2-family survival protein linked to resistance. Turning it down can re-open cell death.

Also appears as: MCL1

Membrane (Cell Membrane)

The cell’s fatty outer layer. Its makeup affects signaling and how drugs get in.

Also appears as: plasma membrane, cell membrane

Metastasis

When cancer spreads to distant places through blood or lymph.

Mevalonate Pathway

The cholesterol/isoprenoid-making route. It supports “prenylation” of proteins like RAS and RHO that cancers use.

Also appears as: mevalonate, HMG-CoA reductase pathway

Microtubules

Protein fibers that pull chromosomes apart during cell division. Some chemo drugs target them.

Also appears as: tubulin

Mito Toxin

A compound that disrupts mitochondria (the cell’s power plants) to stress or kill cancer cells.

Also appears as: mitochondrial toxin, mitotoxin

MMP (Matrix Metalloproteinases)

Scissor-like enzymes that cut the tissue matrix; tumors use them to invade.

Also appears as: MMPs, matrix metalloproteinase

mTOR (Mechanistic Target of Rapamycin)

A major growth-control switch. In many cancers it gets stuck in “grow” mode. mTOR blockers aim to slow cell growth and division.

Also appears as: mTORC1, mTORC2, MTOR

N

Nephro-Protect (Nephroprotective)

Kidney-protective—helps limit drug-related kidney injury.

Also appears as: nephroprotective, renoprotective

Neuropathy

Nerve damage that causes numbness, tingling, or pain—sometimes a side effect of chemotherapy.

NF-κB

A hub for inflammation signals that can help tumor cells survive and resist therapy.

Also appears as: NF-kB, NFκB

NGF (Nerve Growth Factor)

A growth factor that supports nerve survival.

NK Cells (Natural Killer Cells)

Front-line immune cells that can spot and kill abnormal cells—including some cancer cells—without needing prior training.

Also appears as: NK, natural killer cells

NO Donor (Nitric Oxide Donor)

Releases nitric oxide, which can affect blood flow, immune tone, and redox.

Also appears as: NO donor, nitric oxide donor

Nrf2

A control knob for antioxidant defenses. Helpful for normal cells, but if pushed too high in tumors, it may help them cope with stress.

Also appears as: NRF2, NFE2L2, Keap1–Nrf2

O

OXPHOS (Oxidative Phosphorylation)

Mitochondrial energy production. Some tumors lean more on OXPHOS than glycolysis.

Also appears as: oxidative phosphorylation, mitochondrial respiration

P

P-gp (P-glycoprotein)

A drug pump that can spit chemotherapy back out of cancer cells and cause resistance.

Also appears as: ABCB1, MDR1, Pgp, P glycoprotein

p53

A guardian protein that pauses growth or triggers cell death after DNA damage. Often broken in cancer.

Also appears as: TP53

PARP

A DNA repair enzyme. Blocking PARP can exploit certain tumor DNA-repair weaknesses.

Also appears as: poly(ADP-ribose) polymerase

PD-1

A brake on T-cells. When PD-1 meets PD-L1, immune attack slows. Checkpoint drugs lift this brake.

Also appears as: programmed cell death protein 1

PD-L1

A “don’t attack me” signal some tumors show to shut down T-cells. Checkpoint drugs can block it.

Also appears as: programmed death-ligand 1

PDK (Pyruvate Dehydrogenase Kinase)

Shifts metabolism toward glycolysis by turning down the enzyme that feeds mitochondria.

Also appears as: PDK2, PDK3, PDK4, pyruvate dehydrogenase kinase

PDK1 (3-Phosphoinositide-Dependent Protein Kinase-1)

A kinase upstream of AKT in the PI3K pathway (different from the PDKs that act on pyruvate).

Also appears as: PDK-1, PDPK1

Perfusion

Blood flow through tissues. Better perfusion can improve oxygen and drug delivery.

Pharmacodynamics (PD)

What the drug does to the body—how it works at its targets and what effects it causes.

Also appears as: PD

Pharmacokinetics (PK)

What the body does to a drug—absorption, distribution, metabolism, excretion.

Also appears as: PK

PI3K

Relay switch upstream of AKT. Together, the PI3K–AKT–mTOR pathway is a major driver of tumor growth.

Also appears as: PI3K–AKT–mTOR, phosphoinositide 3-kinase

PPAR

A family of nuclear receptors (α/δ/γ) that tune lipid and glucose metabolism and inflammation.

Also appears as: PPAR-alpha, PPAR-delta, PPAR-gamma

Pro-oxidant

Pushes oxidative stress higher (often selectively in tumors at high doses).

Also appears as: prooxidant

Proteasome

The cell’s protein recycler. Blocking it can overwhelm tumor cells and trigger death.

Q

QoL (Quality of Life)

How a person feels and functions day to day during or after treatment.

Also appears as: quality of life, QOL

R

Radiosensitizer

Makes tumor cells easier to damage with radiation.

Also appears as: radiosensitization

Redox (Reduction–Oxidation Balance)

The cell’s see-saw between oxidants (like ROS) and antioxidants (like glutathione). Cancer cells often tilt this balance in their favor, and some therapies exploit that tilt.

Also appears as: redox balance, oxidation–reduction

Redox Cycler

A compound that flips between reduced and oxidized forms, often generating ROS along the way.

Also appears as: redox cycling

Rho (Rho GTPases)

Small switches that control cell shape and movement; can drive invasion and spread.

Also appears as: RHOA, RHOB, RHOC, Rho pathway

ROS (Reactive Oxygen Species)

Short-lived, very reactive oxygen molecules that can damage DNA, proteins, and cell membranes. Tumors often run “hotter” with more ROS. Some treatments deliberately push ROS higher to stress or kill cancer cells.

Also appears as: ROS, reactive oxygen species, oxidative stress

S

Senolytic

A compound that selectively removes old, damaged (senescent) cells.

Sirtuin

A family of stress-response enzymes linked to metabolism and aging.

Also appears as: SIRT1, SIRT2, SIRT3, SIRT

STAT3

A signal-to-gene switch tied to inflammation, survival, and spread (metastasis).

Also appears as: JAK–STAT, STAT

T

T-Cell

Adaptive immune cells (CD4 helpers, CD8 killers) that coordinate and carry out anti-tumor responses.

Also appears as: T cell, T cells, T lymphocyte

Telomere

Protective caps at the ends of chromosomes. Tumors often maintain them to keep dividing.

Also appears as: telomeres, telomerase

Th1 Cytokines

Immune messages (like IFN-γ, IL-2) that support T-cell–driven anti-tumor responses.

Also appears as: Th1, Type 1 cytokines, IFN-γ, IL-2

Thrombolytic

A drug that dissolves clots (for example, plasminogen activators).

Topoisomerase II (Topo II)

A DNA “untangler.” Blocking it (with drugs like anthracyclines) stops proper DNA handling in dividing cells.

Also appears as: Topo-II, TOP2

TRAIL

A natural signal (TNF family) that can trigger death receptors on tumor cells.

Also appears as: TNFSF10

Treg Mod (Regulatory T-cell Modulation)

Reducing or reshaping suppressive T-cells so the immune system can better attack cancer.

Also appears as: Treg modulation, Treg

TrxR (Thioredoxin Reductase)

A redox enzyme that keeps thioredoxin in its active state.

Also appears as: thioredoxin reductase

V

VDR (Vitamin D Receptor)

A gene switch turned on by vitamin D that can influence cell growth and differentiation.

VEGF

A key “grow more blood vessels” signal. Many anti-angiogenic drugs target VEGF.

Also appears as: vascular endothelial growth factor

W

Warburg Effect

Many tumors favor sugar-burning (glycolysis) even when oxygen is available, supporting rapid growth.

Also appears as: aerobic glycolysis

Wnt Pathway

A growth and differentiation pathway often miswired in cancer.

Also appears as: WNT, β-catenin

Β

β-Glucan

Immune-modulating fibers from yeast, oats, or mushrooms that can activate innate immune cells.

Also appears as: B-Glucan, beta-glucan, β glucan

β-Oxidation

How mitochondria break down fats for energy.

Also appears as: B-Oxidation, beta-oxidation

Note: Educational only; not medical advice. Always coordinate care with your licensed clinician.