Research Radartracking 1,138 published studies · 277 human · 6 safety signals · 42 clinical trials · 44 cancer pages · updated Jul 2026Open the Research Map →

Mebendazole †Rx

Repurposed Rx: Tubulin disruptor, VEGF ↓, apoptosis ↑; phase I/II active in glioma/ovarian/colorectal; chemo synergies.

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Human-reviewed · How we review →

AI extractedhuman reviewedsources checkedretractions suppressed

Evidence at a glanceLab onlyReported positive
1 published studies tagged to this agent0 human studies approved & graded (trial, observational, or meta-analysis)
Why this grade?

Lab onlyLab / cell studies only — no human or animal data.

Computed deterministically from the studies’ types and reported outcomes — not written by AI, and not a claim that anything works.

👥⭐⭐⭐ Moderate — Robust preclinical data; phase I/II trials show safety and signals in glioma/ovarian; larger RCTs ongoing.MBZVermoxEmverm

Forms: Oral tablets (100 mg, 500 mg chewable) · Compounded suspension

Educational only, not medical advice. OncoForge makes no claim that Mebendazole †Rx treats, prevents, or cures any condition, beyond what the linked studies show. Evidence levels vary; effects may not translate to people, and some compounds can cause harm. Always coordinate with your oncology team.

Key Takeaway

Anthelmintic repurposed for oncology: Potent tubulin disruptor with anti-angiogenic and pro-apoptotic actions; strong preclinical efficacy and emerging phase I/II signals, particularly in brain and gynecologic cancers.

Evidence at a glance

Tier 2 · animalGliomaOvarianColorectalProstatePancreatic

Extensive in vitro/in vivo validation; phase I/II trials confirm safety/PK and signals in glioma (NCT01729260), ovarian (NCT03925662); synergies with TMZ/cisplatin; ongoing 2025 trials in H&N/pancreatic.

How it may work

Mebendazole (MBZ) inhibits microtubule polymerization by binding β-tubulin, disrupting mitosis and inducing G2/M arrest; suppresses VEGF/HIF-1α signaling for anti-angiogenic effects; activates intrinsic apoptosis via caspase-3/9, Bax upregulation, and p53 stabilization; additional targets include Hedgehog, NF-κB, and kinase pathways; penetrates BBB effectively; preclinical and early clinical data in glioma, ovarian, colorectal, and other solid tumors.

Targets & pathways

Curated mechanistic targets reported for this agent — how it may act on cells, not proof of a clinical effect.

  • TubulinMicrotubule polymerization inhibition → mitotic arrest
  • AngiogenesisVEGF/HIF-1α suppression
  • ApoptosisCaspase activation, p53 stabilization
  • HedgehogSMO inhibition in some models
  • NF-κBInflammation and survival signaling ↓
TubulinAngiogenesisApoptosis

Often studied / combined with

Combinations reported in the literature, not a protocol or a recommendation.

Overlapping mechanisms

Safety & interactions

Severity and how well-established each signal is are shown separately. Verify everything with your oncologist or pharmacist — absence here does not mean safe.

Risk categories
HepatotoxicityGi UpsetNeutropenia
Potential interactions
  • CYP3A4 inducersMonitorModerateTheoreticalReduces MBZ levels (e.g., rifampin, carbamazepine).
  • CYP3A4 inhibitorsCautionModerateTheoreticalIncreases exposure (e.g., ketoconazole).
  • TemozolomideSynergizeLowTheoreticalAdditive BBB penetration and anti-glioma effects.

Timing

References

Research

Where the evidence is

What has been studied, and how strong it is, by topic. A dashed cell means no studies were found for that combination — a gap, not evidence of no effect. Open a row to see its studies.

CancerHuman evidenceMechanismSafetyTrial
Canine High Grade Astrocytoma1
Glioma1

What supports this page

The kinds of sources behind this page, strongest at the top. Faint rungs show what is not here yet.

Guideline
0
Meta-analysis
0
Systematic review
0
Randomized trial
0
Clinical trial
0
Observational
0
Case report
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Review
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Preclinical
1
Other
0
1 studies1 lab

Tracking 1 published study of Mebendazole: 1 in the lab.

Reported direction across studies: 1 positive.

No human studies yet — these are preclinical (lab/animal) findings that may not translate to people.

These counts summarize what the studies reported; they are not a measure of whether Mebendazole works.

Cancers named in these studies

canine high-grade astrocytoma (1)glioma (1)

All studies

Lab · in vitroReported positivePreclinical onlyTier 1 · lab

European Mistletoe (Viscum album) Extract Is Cytotoxic to Canine High-Grade Astrocytoma Cells In Vitro and Has Additive Effects with Mebendazole

Veterinary sciences · Jan 2022 · in vitro dose-response and combination assays using the canine SDT-3G high-grade astrocytoma cell line

Mebendazolecanine high-grade astrocytomaglioma

This laboratory study tested European mistletoe (Viscum album) extract on a canine high-grade astrocytoma cell line (SDT-3G) and measured effects alone and combined with mebendazole. Mistletoe extract had an IC50 of 5.644 ± 0.09 SD µg/mL in these cells, and combining mistletoe (5 µg/mL) with mebendazole (0.03 µM) increased cell death compared with each drug alone. The authors conclude the results support further in vitro and in vivo study in dogs.

Reported effects: IC50 mistletoe 5.644 · IC50 mebendazole 0.03 · +1 more

Studied with: mebendazole.

Key findings
  • The IC50 for mistletoe alone was 5.644 ± 0.09 SD µg/mL against SDT-3G cells in vitro.
  • Mebendazole was applied at a previously determined IC50 of 0.03 µM in combination experiments.
  • The addition of mistletoe at 5 µg/mL to mebendazole at 0.03 µM led to increased cell death compared to what would be expected for each drug separately.
Limitations: In vitro study only (cell line); no in vivo or clinical data.; Single canine glioma cell line (SDT-3G) used — limited generalizability across tumors.; Abstract does not report sample size, replicate numbers, or statistical test results for the combination effect.; No detailed mechanistic investigation reported in the abstract.; No safety, pharmacokinetics, or efficacy data in animals or humans..

AI summary of the abstract, human-reviewed · Jul 2026. Describes what this study reported, not medical advice. View on PubMed · Full text

What changed recently

The latest additions to Mebendazole †Rx's evidence base, and anything that's been retracted.

Recently added

Cancers where Mebendazole †Rx reported positive results

Where at least one study reported a positive result, shown with the full picture, not just the wins. Positive results are more likely to be published, and most of these are early lab or animal studies that may not translate to people. This reports what studies found, not what works.

Preclinical only: lab / animal (2)
Canine high-grade astrocytoma1 positive1 lab
Limitations: In vitro study only (cell line); no in vivo or clinical data.; Single canine glioma cell line (SDT-3G) used — limited generalizability across tumors.; Abstract does not report sample size, replicate numbers, or statistical test results for the combination effect.; No detailed mechanistic investigation reported in the abstract.; No safety, pharmacokinetics, or efficacy data in animals or humans..
Cited positive studies (1)
Glioma1 positive1 lab
Limitations: In vitro study only (cell line); no in vivo or clinical data.; Single canine glioma cell line (SDT-3G) used — limited generalizability across tumors.; Abstract does not report sample size, replicate numbers, or statistical test results for the combination effect.; No detailed mechanistic investigation reported in the abstract.; No safety, pharmacokinetics, or efficacy data in animals or humans..
Cited positive studies (1)

Evidence at a glance: Mebendazole †Rx by cancer

A deterministic grade of what published studies report for each: strength of evidence, the reported direction, and the largest credible effect, strongest-evidence first. This summarizes findings; it is not a claim that anything works.

Canine high-grade astrocytomaLab onlyReported positive1 lab

Lab / cell studies only — no human or animal data.

Largest credible effect: IC50 mistletoe 5.644 PMID 35051115 · effect sizes 0.03–5.644 across 2 studies

Most authoritative study: European Mistletoe (Viscum album) Extract Is Cytotoxic to Canine High-Grade Astrocytoma Cells In Vitro and Has Additive Effects with Mebendazole

No human studies yet · Based on a single study.
GliomaLab onlyReported positive1 lab

Lab / cell studies only — no human or animal data.

Largest credible effect: IC50 mistletoe 5.644 PMID 35051115 · effect sizes 0.03–5.644 across 2 studies

Most authoritative study: European Mistletoe (Viscum album) Extract Is Cytotoxic to Canine High-Grade Astrocytoma Cells In Vitro and Has Additive Effects with Mebendazole

No human studies yet · Based on a single study.

Dose: as studied, not a recommendation

These are doses as studied or reported, never a recommendation. The right amount of Mebendazole †Rx depends on you, your other medicines, and your situation; decide it with your oncology team and pharmacist, not from a web page.

Ranges seen in adjunct / practice use: 100–1500 mg/day (po) divided BID-TID; with fatty meal for absorption, Anti-parasitic 100 mg BID; oncology trials 200-500 mg BID (up to 1500 mg/day in glioma); fatty food increases bioavailability 2-3x..

Doses reported in studies

Trials studying Mebendazole †Rx

No actively-recruiting trials matched right now. Recruiting is not the same as proven. Search ClinicalTrials.gov →

Appears in these protocol claims

Mebendazole †Rx is named in these protocols discussed online. Listed for transparency: being part of a protocol is not evidence that it works, and OncoForge does not endorse them.

Inclusion here is not an endorsement. OncoForge makes no claim beyond what the linked studies show. Discuss anything on this page with your oncology team before acting on it.

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